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262-0203-00L 1 Credits DR , MSC D-INFK , D-BSSE

Computer-Assisted Drug Design (CADD) Essentials

VVZ CR n/a

Last Updated: 2026-06-03 00:07:32

Abstract

This course introduces the concepts of computer-aided drug discovery (CADD) and design, covering essential techniques like compound library analysis, virtual screening, de novo molecular design and optimisation. Through practical exercises, participants will learn to use software and prediction models to identify and optimise bioactive molecules.

Objective

Participants learn to (i) analyse and interpret the output of CADD software; (ii) evaluate the quality of virtual screening hits and computer-generated molecules; (iii) assess the predictive power of models; and (iv) translate results into actionable insights.

Content

The course equips participants with the knowledge to understand and effectively utilise computational approaches in the early drug discovery process. Participants will learn essential concepts of molecular representation and interaction, cheminformatics, ligand- and structure-based molecular design, molecular modeling, property prediction, and applied artificial intelligence in drug discovery.

Resources

Lecture Notes

Accompanying lecture slides are provided.

Literature

G. Klebe: «Drug Design», Springer, 2024. G. Schneider, K.-H. Baringhaus: «Molecular Design - Concepts and Applications», Wiley-VCH, 2008.

General Information

Language
English
Levels
DR , MSC
Frequency
Yearly recurring

Examination

Type
ungraded semester performance
Exercises and oral report during the course

Registration & Places

Max Places
20
Signup End
11.10.2026

Course Components

Type Title Time & Place Hours
lecture with exercise Computer-Assisted Drug Design (CADD) Essentials
Block Course: 8-10 September 2026 (all day) The course takes place in person at D-BSSE in BASEL
No time listed 24 h semesterly

Offered In